A new paradigm for protein kinase inhibition : blocking phosphorylation without directly targeting ATP bindingBOGOYEVITCH, Marie A; FAIRLIE, David P.Drug discovery today. 2007, Vol 12, Num 15-16, pp 622-633, issn 1359-6446, 12 p.Article

Nonpeptide ligands that target peptide-activated GPCRs in inflammationBLAKENEY, Jade S; FAIRLIE, David P.Current medicinal chemistry. 2005, Vol 12, Num 25, pp 3027-3042, issn 0929-8673, 16 p.Article

Synthesis of the Thiazole―Thiazoline Fragment of Largazole AnaloguesDINESS, Frederik; NIELSEN, Daniel S; FAIRLIE, David P et al.Journal of organic chemistry. 2011, Vol 76, Num 23, pp 9845-9851, issn 0022-3263, 7 p.Article

Macrocycles mimic the extended peptide conformation recognized by aspartic, serine, cysteine and metallo proteasesTYNDALL, Joel D. A; FAIRLIE, David P.Current medicinal chemistry. 2001, Vol 8, Num 8, pp 893-907, issn 0929-8673Article

Matching Cavities in G Protein-Coupled Receptors to Infer Ligand-Binding SitesMADALA, Praveen K; FAIRLIE, David P; BODEN, Mikael et al.Journal of chemical information and modeling. 2012, Vol 52, Num 5, pp 1401-1410, issn 1549-9596, 10 p.Article

Therapeutic targets in inflammatory diseaseHUME, David A; FAIRLIE, David P.Current medicinal chemistry. 2005, Vol 12, Num 25, pp 2925-2929, issn 0929-8673Article

MR1 presents microbial vitamin B metabolites to MAIT cellsKJER-NIELSEN, Lars; PATEL, Onisha; WILLIAMSON, Nicholas A et al.Nature (London). 2012, Vol 491, Num 7426, pp 717-723, issn 0028-0836, 7 p.Article

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A convergent solution-phase synthesis of the macrocycle Ac-Phe-[Orn-Pro-D-Cha-Trp-Arg], a potent new antiinflammatory drugREID, Robert C; ABBENANTE, Giovanni; TAYLOR, Stephen M et al.Journal of organic chemistry. 2003, Vol 68, Num 11, pp 4464-4471, issn 0022-3263, 8 p.Article

Towards Histone Deacetylase Inhibitors as New Antimalarial DrugsANDREWS, Katherine T; TRAN, Thanh N; FAIRLIE, David P et al.Current pharmaceutical design (Print). 2012, Vol 18, Num 24, pp 3467-3479, issn 1381-6128, 13 p.Article

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Structures of peptide agonists for human protease activated receptor 2STOERMER, Martin J; FLANAGAN, Bernadine; BEYER, Renee L et al.Bioorganic & medicinal chemistry letters (Print). 2012, Vol 22, Num 2, pp 916-919, issn 0960-894X, 4 p.Article

Mutagenesis of the West Nile virus NS2B cofactor domain reveals two regions essential for protease activityCHAPPELL, Keith J; STOERMER, Martin J; FAIRLIE, David P et al.Journal of general virology. 2008, Vol 89, pp 1010-1014, issn 0022-1317, 5 p., 4Article

Single turn peptide alpha helices with exceptional stability in waterSHEPHERD, Nicholas E; HOANG, Huy N; ABBENANTE, Giovanni et al.Journal of the American Chemical Society. 2005, Vol 127, Num 9, pp 2974-2983, issn 0002-7863, 10 p.Article

Conformationally homogeneous cyclic tetrapeptides: Useful new three-dimensional scaffoldsGLENN, Matthew P; KELSO, Michael J; TYNDALL, Joel D. A et al.Journal of the American Chemical Society. 2003, Vol 125, Num 3, pp 640-641, issn 0002-7863, 2 p.Article

Metal clips induce folding of a Short unstructured peptide into an α-helix via turn conformations in water. Kinetic versus thermodynamic productsBEYER, Renée L; HOANG, Huy N; APPLETON, Trevor G et al.Journal of the American Chemical Society. 2004, Vol 126, Num 46, pp 15096-15105, issn 0002-7863, 10 p.Article

Conformationally constrained macrocycles that mimic tripeptide β-strands in water and aprotic solventsREID, Robert C; KELSO, Michael J; SCANLON, Martin J et al.Journal of the American Chemical Society. 2002, Vol 124, Num 20, pp 5673-5683, issn 0002-7863Article

Folding pentapeptides into left and right handed alpha helicesHOANG, Huy N; ABBENANTE, Giovanni; HILL, Timothy A et al.Tetrahedron (Oxford. Print). 2012, Vol 68, Num 23, issn 0040-4020, 4335, 4513-4516 [5 p.]Article

Ex Vivo Activity of Histone Deacetylase Inhibitors against Multidrug-Resistant Clinical Isolates of Plasmodium falciparum and P. vivaxMARFURT, Jutta; CHALFEIN, Ferryanto; PRICE, Ric N et al.Antimicrobial agents and chemotherapy. 2011, Vol 55, Num 3, pp 961-966, issn 0066-4804, 6 p.Article

Inhibitors selective for HDAC6 in enzymes and cellsGUPTA, Praveer K; REID, Robert C; LIGONG LIU et al.Bioorganic & medicinal chemistry letters (Print). 2010, Vol 20, Num 23, pp 7067-7070, issn 0960-894X, 4 p.Article

Antiproliferative and phenotype-transforming antitumor agents derived from cysteineGLENN, Matthew P; KAHNBERG, Pia; BOYLE, Glen M et al.Journal of medicinal chemistry (Print). 2004, Vol 47, Num 12, pp 2984-2994, issn 0022-2623, 11 p.Article

Protective effect of a new C5a receptor antagonist against ischemia-reperfusion injury in the rat small intestineARUMUGAM, Thiruma V; SHIELS, Ian A; WOODRUFF, Trent M et al.The Journal of surgical research. 2002, Vol 103, Num 2, pp 260-267, issn 0022-4804Article